Product Description:
CAS: 41354-29-4
MF: C21H22ClN
MW: 323.86
EINECS: 213-535-1
Product Categories: Building Blocks;Heterocyclic Building Blocks;Piperidines;API;PERIACTIN
Melting point:165 °C (dec.)(lit.)
Solubility Ethanol :soluble
Appearance:Off white powders
Usage:H1-antihistamine, antipruriticÂ
Usage:
Cyproheptadine is a first-generation antihistamine with additional anticholinergic, antiserotonergic, and local anesthetic properties.Cyproheptadine is a 5-HT2/5-HT1C serotonin receptor antagonist; H 1 histamine receptor antagonist; antipruritic .Â
Antihistamines:Â
1.Cyproheptadine hydrochloride is a kind of pipecolic antihistamines,it can compete with histamine released from the organization for H1 receptor on effector cells , thereby it can prevent the onset of an allergic reaction, and release histamine-induced spasm and congestion effects, this product has a strong H1 receptor antagonism, its anti-histamine effect is stronger than chlorpheniramine, promethazine . There are mild to moderate anti-serotonin effects and anticholinergic effects. In addition, there is a stimulate appetite effect, and weight gains after a certain time.Â
2.Clinically cyproheptadine hydrochloride is mainly used for acute and chronic urticaria (especially it has a good effect on cold urticaria ), papular urticaria, angioedema, atopic eczema, contact dermatitis, food allergy, drug allergy, allergic rhinitis, hay fever, allergic conjunctivitis, allergic to insect stings and migraine. It has some therapeutic effect on bronchial asthma . It is acceptable for the adjuvant treatment of Cushing's syndrome, acromegaly. In addition,as an appetite enhancer,it is used for neuropathic fear of food. There are reports about acanthosis nigricans treatment, prevention of necrotizing pyoderma.
3.Dosage oral often release dosage : (1) allergic diseases: adult, once 2 ~ 4mg, one day 2 or 3 times. (2) Cushing's syndrome, applicable to the treatment of cases of bilateral adrenal hyperplasia,it can inhibit the hypothalamic release of corticotropin releasing hormone (CRH) and inhibit the secretion of pituitary adrenocorticotropic hormone (ACTH), thereby lowering plasma ACTH and cortisol levels; adults start one day 8mg,which can be gradually increased to one day24mg; the usual dose is one day 12 ~ 24mg, divided doses,it needs long-term use; in the case of cortical function inadequate after total resection or subtotal bilateral adrenal, on one hand ,supple corticosteroids, on the other hand,take cyproheptadine,which can reduce the chance of occurrence of pituitary tumors .
Cyproheptadine Hydrochloride Uses:
Anticoagulant, anti-allergic drugs. It can be used for urticaria, eczema, and allergic contact dermatitis, skin itching and other allergic reactions. It can also be used for Cushing's diseases and acromegaly . Â
Sulbutiamine CAS 3286-46-2
Aniracetam CAS 72432-10-1
Noopept CAS 157115-85-0
Idra-21 CAS 22503-72-6
4-Aminobutyric acid CAS 56-12-2
NSI-189 Free Base CAS 1270138-40-3
NSI-189 Phosphate CAS 1270138-41-4
9-fluorenol CAS 1689-64-1
Coluracetam CAS 135463-81-9
Sunifiram CAS 314728-85-3
Pramiracetam CAS 68497-62-1
Piracetam CAS 7491-74-9
Oxiracetam CAS 62613-82-5
Fasoracetam CAS 110958-19-5
Nefiracetam CAS 77191-36-7
Centrophenoxine CAS 3685-84-5
Pikamilon Sodium CAS 62936-56-5
PRL-8-53 HCL CAS : 51352-87-5
Meclofenoxate hydrochloride CAS:3685-84-5
Levodopa(L-DOPA) CAS:59-92-7
Etiracetam(UCB-6474) CAS:33996-58-6
Product Description:
CAS: 41354-29-4
MF: C21H22ClN
MW: 323.86
EINECS: 213-535-1
Product Categories: Building Blocks;Heterocyclic Building Blocks;Piperidines;API;PERIACTIN
Melting point:165 °C (dec.)(lit.)
Solubility Ethanol :soluble
Appearance:Off white powders
Usage:H1-antihistamine, antipruriticÂ
Usage:
Cyproheptadine is a first-generation antihistamine with additional anticholinergic, antiserotonergic, and local anesthetic properties.Cyproheptadine is a 5-HT2/5-HT1C serotonin receptor antagonist; H 1 histamine receptor antagonist; antipruritic .Â
Antihistamines:Â
1.Cyproheptadine hydrochloride is a kind of pipecolic antihistamines,it can compete with histamine released from the organization for H1 receptor on effector cells , thereby it can prevent the onset of an allergic reaction, and release histamine-induced spasm and congestion effects, this product has a strong H1 receptor antagonism, its anti-histamine effect is stronger than chlorpheniramine, promethazine . There are mild to moderate anti-serotonin effects and anticholinergic effects. In addition, there is a stimulate appetite effect, and weight gains after a certain time.Â
2.Clinically cyproheptadine hydrochloride is mainly used for acute and chronic urticaria (especially it has a good effect on cold urticaria ), papular urticaria, angioedema, atopic eczema, contact dermatitis, food allergy, drug allergy, allergic rhinitis, hay fever, allergic conjunctivitis, allergic to insect stings and migraine. It has some therapeutic effect on bronchial asthma . It is acceptable for the adjuvant treatment of Cushing's syndrome, acromegaly. In addition,as an appetite enhancer,it is used for neuropathic fear of food. There are reports about acanthosis nigricans treatment, prevention of necrotizing pyoderma.
3.Dosage oral often release dosage : (1) allergic diseases: adult, once 2 ~ 4mg, one day 2 or 3 times. (2) Cushing's syndrome, applicable to the treatment of cases of bilateral adrenal hyperplasia,it can inhibit the hypothalamic release of corticotropin releasing hormone (CRH) and inhibit the secretion of pituitary adrenocorticotropic hormone (ACTH), thereby lowering plasma ACTH and cortisol levels; adults start one day 8mg,which can be gradually increased to one day24mg; the usual dose is one day 12 ~ 24mg, divided doses,it needs long-term use; in the case of cortical function inadequate after total resection or subtotal bilateral adrenal, on one hand ,supple corticosteroids, on the other hand,take cyproheptadine,which can reduce the chance of occurrence of pituitary tumors .
Cyproheptadine Hydrochloride Uses:
Anticoagulant, anti-allergic drugs. It can be used for urticaria, eczema, and allergic contact dermatitis, skin itching and other allergic reactions. It can also be used for Cushing's diseases and acromegaly . Â
Sulbutiamine CAS 3286-46-2
Aniracetam CAS 72432-10-1
Noopept CAS 157115-85-0
Idra-21 CAS 22503-72-6
4-Aminobutyric acid CAS 56-12-2
NSI-189 Free Base CAS 1270138-40-3
NSI-189 Phosphate CAS 1270138-41-4
9-fluorenol CAS 1689-64-1
Coluracetam CAS 135463-81-9
Sunifiram CAS 314728-85-3
Pramiracetam CAS 68497-62-1
Piracetam CAS 7491-74-9
Oxiracetam CAS 62613-82-5
Fasoracetam CAS 110958-19-5
Nefiracetam CAS 77191-36-7
Centrophenoxine CAS 3685-84-5
Pikamilon Sodium CAS 62936-56-5
PRL-8-53 HCL CAS : 51352-87-5
Meclofenoxate hydrochloride CAS:3685-84-5
Levodopa(L-DOPA) CAS:59-92-7
Etiracetam(UCB-6474) CAS:33996-58-6
Antihistamines Pharmaceutical Raw Materials Cyproheptadine Hydrochloride CAS 41354-29-4
Model NO.: 41354-29-4
Leading Time: Within 12hours Ater Payment
Delivery Time: 3-5working Days After Payment
Melting Point: 81-82c
Density: 1.08 g/cm3
Flash Point: 469.7 C at 760 Mmhg
Heavy Metals: Max.0.001%
Storage: Cool and Dry
Related Compound E: Max. 0.1%
Limit of Cyclohexane: Max. 0.08%
Individual Unspecified Impurlty: Max. 0.1%
Trademark: ZJY
Transport Package: Discreet Package
Specification: White Powder
Origin: China
HS Code: 30013006
Model NO.: 41354-29-4
Leading Time: Within 12hours Ater Payment
Delivery Time: 3-5working Days After Payment
Melting Point: 81-82c
Density: 1.08 g/cm3
Flash Point: 469.7 C at 760 Mmhg
Heavy Metals: Max.0.001%
Storage: Cool and Dry
Related Compound E: Max. 0.1%
Limit of Cyclohexane: Max. 0.08%
Individual Unspecified Impurlty: Max. 0.1%
Trademark: ZJY
Transport Package: Discreet Package
Specification: White Powder
Origin: China
HS Code: 30013006